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TG4-155

Catalogue number:
CAY17639-10 mg
Supplier:
Size:
10 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£142.00 Estimated delivery Fri 9 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1164462-05-8

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

394.5

Alternative Names:

(2e)-n-[2-(2-methyl-1h-indol-1-yl)ethyl]-3-(3,4,5-trimethoxyphenyl)-2-propenamide

Product Description:

A selective, brain penetrant EP2 antagonist (KB = 2.4 nM); blocks the induced expression of inflammatory markers in microglial cells treated with butaprost; reduces neurodegeneration in a mouse model of status epilepticus; inhibits proliferation and invasion in cancer cells treated with butaprost

Storage Temperature:

-20°C

CAY17639-10 mg: TG4-155
CAY17639-10 mg: TG4-155
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