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Mps1-IN-2

Catalogue number:
CAY19401-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£42.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1228817-38-6

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

480.6

Alternative Names:

9-cyclopentyl-2-[[2-ethoxy-4-(4-hydroxy-1-piperidinyl)phenyl]amino]-5,7,8,9-tetrahydro-5-methyl-6h-pyrimido[4,5-b][1,4]diazepin-6-one

Product Description:

An inhibitor of Mps1 (IC50 = 145 nM); 1,000-fold selective for Mps1 over a panel of 352 kinases at 10 mM, but does inhibit Plk1 (Kd = 61 nM)

Storage Temperature:

-20°C

CAY19401-1 mg: Mps1-IN-2
CAY19401-1 mg: Mps1-IN-2
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