BMX-IN-1
Catalogue number:
CAY19165-500 ug
Supplier:
Size:
500 µg
Product is available in:
£54.00
Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1431525-23-3
Purity:
≥95%
Formulation:
A crystalline solid
Molecular Weight:
524.6
Alternative Names:
n-[2-methyl-5-[9-[4-[(methylsulfonyl)amino]phenyl]-2-oxobenzo[h]-1,6-naphthyridin-1(2h)-yl]phenyl]-2-propenamide, bmx inhibitor 1
- Data sheet: View or download
- MSDS: View or download
Product Description:
An irreversible inhibitor of BMX (IC50 = 8 nM) and BTK (IC50 = 10.4 nM); inhibits the proliferation of Tel-BMX-transformed Ba/F3 prostate cancer cells (GI50 = 25 nM), as well as RV-1, DU-145, PC-3, and VCAP prostate cancer cell lines (GI50s = 2.54, 4.38, 5.37, and 2.46 µM, respectively)
Storage Temperature:
-20°C
