Fluspirilene
Catalogue number:
CAY19530-5 mg
Supplier:
Size:
5 mg
Product is available in:
£94.00
Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1841-19-6
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Weight:
475.6
Alternative Names:
8-[4,4-bis(4-fluorophenyl)butyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one, mcn-jr 6218, r 6218, redeptin
- Data sheet: View or download
- MSDS: View or download
Product Description:
A dopamine D2 and D3 receptor antagonist (Kis = 1.5 and 1.1 nM, respectively); selective for dopamine D2 and D3 receptors over dopamine D1, α1- and α2-adrenergic, H1 histamine, and σ1 receptors (Kis = 450, 102, >5,000, 540, and 150 nM, respectively), mAChRs (Ki = >5,000 nM), and 5-HT1A, 5-HT1B, 5-HT2C, and 5-HT3 receptors (Kis = 110, >5,000, 1,830, and >5,000 nM, respectively); noncompetitive inhibitor of Cav1 channels (IC50 = 30 nM); inhibits apomorphine-induced vomiting in dogs (ED50 = 0.011 mg/kg)
Storage Temperature:
-20°C
