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Glutaminase Inhibitor Compound 968

Catalogue number:
CAY17199-10 mg
Supplier:
Size:
10 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£159.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

311795-38-7

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

475.4

Alternative Names:

5-[3-bromo-4-(dimethylamino)phenyl]-2,3,5,6-tetrahydro-2,2-dimethyl-benzo[a]phenanthridin-4(1h)-one

Product Description:

A cell-permeable, reversible inhibitor of a mitochondrial glutaminase splice variant, glutaminase C (IC50 = ~2.5 µM), which is commonly found in cancer cells; blocks transformation induced by Rho GTPases and inhibits the proliferation of cancer cell lines without affecting normal cells

Storage Temperature:

-20°C

CAY17199-10 mg: Glutaminase Inhibitor Co
CAY17199-10 mg: Glutaminase Inhibitor Compound 968
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