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GW 803430

Catalogue number:
CAY13948-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£58.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

515141-51-2

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

482

Alternative Names:

6-(4-chlorophenyl)-3-[3-methoxy-4-[2-(1-pyrrolidinyl)ethoxy]phenyl]-thieno[3,2-d]pyrimidin-4(3h)-one, gw 3430

Product Description:

An antagonist of MCH1 (IC50 = 0.5 nM); reduces cumulative body weight and food intake in diet-induced obese rats at 1 and 3 mg/kg; decreases marble-burying behavior in mice without affecting performance in the rotorod test at 10 and 30 mg/kg; reduces immobility time in the forced swim and tail suspension tests in mice at 3 and 10 mg/kg, respectively

Storage Temperature:

-20°C

CAY13948-1 mg: GW 803430
CAY13948-1 mg: GW 803430
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