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LJI308

Catalogue number:
CAY19924-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£251.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1627709-94-7

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

368.4

Alternative Names:

2,6-difluoro-4-[4-[4-(4-morpholinyl)phenyl]-3-pyridinyl]-phenol

Product Description:

A selective and potent inhibitor of RSKs (IC50 = 4-13 nM for RSK isoforms 1-3); reduces phosphorylation of YB1 in MDA-MB-231 cells bearing activating mutations in the MAPK signaling pathway (EC50 = 0.21 µM); reduces H358 growth in soft agar and colony forming assays.

Storage Temperature:

-20°C

CAY19924-5 mg: LJI308
CAY19924-5 mg: LJI308
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