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AZD 3965

Catalogue number:
CAY19912-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£63.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1448671-31-5

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

515.5

Alternative Names:

5-[[(4s)-4-hydroxy-4-methyl-2-isoxazolidinyl]carbonyl]-3-methyl-1-(1-methylethyl)-6-[[5-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]methyl]-thieno[2,3-d]pyrimidine-2,4(1h,3h)-dione

Product Description:

A selective inhibitor of MCT1 (Ki = 1.6 nM), killing tumor cells that are reliant on glycolysis by blocking lactate transport; increases intratumor lactate levels and decreases tumor growth in mice bearing SCLC xenografts

Storage Temperature:

-20°C

CAY19912-1 mg: AZD 3965
CAY19912-1 mg: AZD 3965
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