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CGP 57380

Catalogue number:
CAY13322-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£142.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

522629-08-9

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

244.2

Alternative Names:

n3-(4-fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidine-3,4-diamine, mnk1 inhibitor

Product Description:

A selective inhibitor of MNK1 in vitro (IC50 = 2.2 µM), with no inhibitory activity against p38, JNK1, ERK1/2, PKC, or Src-like kinases; blocks the phosphorylation of eIF4E in response to TNF-α, arsenite, anisomycin, PMA, or fetal calf serum in 293 cells (IC50 = 3 µM)

Storage Temperature:

-20°C

CAY13322-5 mg: CGP 57380
CAY13322-5 mg: CGP 57380
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