Cytisine
Catalogue number:
CAY26437-500 mg
Supplier:
Size:
500 mg
Product is available in:
£532.00
Estimated delivery Fri 9 Aug
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
485-35-8
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Weight:
190.2
Alternative Names:
(1r,5s)-1,2,3,4,5,6-hexahydro-1,5-methano-8h-pyrido[1,2-a][1,5]diazocin-8-one, baptitoxine, cytiton, laburnin, sophorine, tsitafat
- Data sheet: View or download
- MSDS: View or download
Product Description:
An alkaloid and a partial agonist of nAChRs (EC50 = 1 µM for α4β2 subunit-containing nAChRs expressed in Xenopus oocytes); inhibits current induced by acetylcholine by 50% in Xenopus oocytes expressing α4β2-subunit containing nAChRs at 20 nM; binds to α2β2, α2β4, α3β2, α3β4, α4β2, and α4β4 nAChR subunits (Kis = 1.1, 5.4, 37, 220, 1.5, and 2.1 nM, respectively); reduces increases in the ICSS threshold of nicotine-withdrawing rats at 3 mg/kg
Storage Temperature:
-20°C
