This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
249296-44-4
Purity:
99.98
Molecular Weight:
211.26
Alternative Names:
CP 526555
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Varenicline (CP 526555) is a potent partial agonist for α4β2 nicotinic acetylcholine receptor (nAChR) with an EC50 value of 2.3 µM. Varenicline is a full agonist for α3β4 and α7 nAChRs with EC50 values of 55 µM and 18 µM, respectively[2]. Varenicline is a nicotinic ligand based on the structure of cytosine, and has the potential for smoking cessation treatment[5].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)
