This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1888305-96-1
Purity:
98.97
Molecular Formula:
C17H11BrFN3O2
Molecular Weight:
388.19
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
ERK5-IN-2 is an orally active, sub-micromolar, selective ERK5 inhibitor with IC50s of 0.82 µM, 3 µM for ERK5 and ERK5 MEF2D, respectively. ERK5-IN-2 does not interact with the BRD4 bromodomain. ERK5-IN-2 suppresses both tumor xenograft growth and basic fibroblast growth factor (bFGF) driven Matrigel plug angiogenesis[1].
Storage Temperature:
4°C (Powder, protect from light)
