Timapiprant (sodium)
Catalogue number:
HY-15342A-10mg
Supplier:
Size:
10 mg _$$_
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
950688-14-9
Purity:
99.61
Molecular Formula:
C21H16FN2NaO2
Molecular Weight:
370.35
Alternative Names:
OC000459 (sodium)
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Timapiprant sodium (OC000459 sodium) is a potent, selective, and orally active D prostanoid receptor 2 (DP2, also known as CRTH2) antagonist. Timapiprant sodium (OC000459 sodium) potently displaces [3H] PGD2 from human recombinant DP2 (Ki=13 nM), rat recombinant DP2 (Ki=3 nM), and human native DP2 (Ki=4 nM). Timapiprant sodium (OC000459 sodium) inhibits mast cell activation of Th2 lymphocytes and eosinophils[1].
Storage Temperature:
4°C (Powder, stored under nitrogen)
