This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
369631-68-5
Purity:
99.4
Molecular Formula:
C11H6F3NO4
Molecular Weight:
273.16
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Bragsin1 is a potent, selective and noncompetitive inhibitor of the ArfGEF BRAG2, inhibits Arf GTPase activation, with an IC50 of 3 µM. Bragsin1 binds to PH domain of BRAG2, and is a noncompetitive interfacial inhibitor. Bragsin1 has no effect on the Sec7 domain of human ArfGEFs. Anti-cancer activity[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)
