This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1542135-76-1
Purity:
99.43
Molecular Formula:
C19H29N5O3
Molecular Weight:
375.47
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
LML134 (compound 18b) is an orally active and high selective Histamine 3 receptor (H3R) inverse agonist with Kis of 0.3 nM and 12 nM for hH3R cAMP and hH3R bdg. LML134 penetrates the brain rapidly, leading to high H3R occupancy, and disengages its target with a fast kinetic profile. LML134 has the potential for excessive sleep disorders[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)
