This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1454808-95-7
Purity:
98.21
Molecular Formula:
C21H26N6O3
Molecular Weight:
410.47
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
LP-922761 is a potent, selective and orally active adapter protein-2 associated kinase 1 (AAK1) inhibitor with IC50s of 4.8 nM and 7.6 nM in enzyme and cell assays, respectively. LP-922761 also inhibits BMP-2-inducible protein kinase (BIKE) with an IC50 of 24 nM. LP-922761 exhibits no significant activity at cyclin G-associated kinase (GAK), opioid, adrenergic α2 or GABAa receptors[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)