Nebentan (potassium)
Catalogue number:
HY-106994A-5mg
Supplier:
Size:
5 mg _$$_
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
342005-82-7
Purity:
99.53
Molecular Formula:
C24H20KN5O5S
Molecular Weight:
529.61
Alternative Names:
YM598
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Nebentan potassium (YM598) is a potent, selective and orally active non-peptide endothelin ETA receptor antagonist through the modification of Bosentan (HY-A0013). Nebentan potassium inhibits [125I] endothelin-1 binding to cloned human endothelin ETA and ETB receptor, with Ki of 0.697 nM and 569 nM, respectively[1]. YM598 can ameliorate the progression of cor pulmonale and myocardial infarction in vivo[2].
Storage Temperature:
4°C (Powder, sealed storage, away from moisture)