ERRα antagonist-1
Catalogue number:
HY-113960-1ml
Supplier:
Size:
1 ml _$$_
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1072145-33-5
Purity:
98.48
Molecular Formula:
C21H19N3S2
Molecular Weight:
377.53
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
ERRα antagonist-1 (Compound A) is a selective and high affinity estrogen-related receptor α (ERRα) antagonist. ERRα antagonist-1 inhibits interaction of ERRα with Proliferator-activated Receptor γ Coactivator-1α (PGC-1α) and PGC-1β, the IC50 values are 170 nM and 180 nM, respectively. ERRα antagonist-1 does not inhibit the interaction of either ERRβ or ERRγ with PGC-1α and PGC-1β coactivator, and also does not inhibit interaction of ERα or ERβ with PGC-1α or SRC-1[1].
Storage Temperature:
4°C (Powder, protect from light)