This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2804039-78-7
Purity:
98.06
Molecular Formula:
C30H29F3N6O3
Molecular Weight:
578.58
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
GZD856 formic is a potent and orally active PDGFRα/β inhibitor, with IC50s of 68.6 and 136.6 nM, respectively. GZD856 formic is also a Bcr-AblT315I inhibitor, with IC50s of 19.9 and 15.4?nM for native Bcr-Abl and the T315I mutant. GZD856 formic has antitumor activity[1][2]. GZD856 (formic) is a click chemistry reagent, itcontains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
Storage Temperature:
-20°C (Powder, sealed storage, away from moisture)