This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1997369-78-4
Purity:
99.6
Molecular Weight:
527.61
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
GSK8814 is a potent, selective, and ATAD2/2B bromodomain chemical probe and inhibitor, with a binding constant pKd=8.1 and a pKi=8.9 in BROMOscan. GSK8814 binds to ATAD2 and BRD4 BD1 with pIC50s of 7.3 and 4.6, respectively. GSK8814 shows 500-fold selectivity for ATAD2 over BRD4 BD1[1].
Storage Temperature:
-20°C, 3 years (Powder)