£131.00
Estimated delivery Wed 7 Aug
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
864864-17-5
Purity:
≥90%
Formulation:
A solid
Molecular Weight:
349.4
Alternative Names:
2-cyclopropyl-5-[1-(2-fluoro-3-pyridinyl)-5-methyl-1h-1,2,3-triazol-4-yl]-2,3-dihydro-1h-isoindol-1-one
- Data sheet: View or download
- MSDS: View or download
Product Description:
A mGluR1 allosteric antagonist (IC50 = 2.6 nM in CHO cells expressing the human receptor); is selective for mGluR1 over mGluR5 by >2,000-fold, as well as mGluR2, -4, -6, -7, or -8 at 10 µM in CHO cells expressing the human receptors; reduces methamphetamine-induced hyperlocomotion in mice at 1-10 mg/kg, p.o.
Storage Temperature:
-20°C