This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1771691-34-9
Purity:
99.92
Molecular Formula:
C22H18D3FN6O3
Molecular Weight:
439.46
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
BMS-986202 is a potent, selective and orally active Tyk2 inhibitor that binds to Tyk2 JH2 with an IC50 value of 0.19 nM and a Ki of 0.02 nM. BMS-986202 is remarkably selective over other kinases including Jak family members. BMS-986202 is also a weak inhibitor of CYP2C19 with an IC50 value of 14 µM. BMS-986202 can be used for IL-23-driven acanthosis, anti-CD40-induced colitis, and spontaneous lupus research. BMS-986202 is a de novo deuterium[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)