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HA-1077

Catalogue number:
Supplier:
Size:
250 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£341.00 Shipping is calculated in checkout
CAS Number:

203911-27-7

Purity:

≥99%

Molecular Weight:

364.3

Product Description:

Dihydrochloride form of HA-1077. Inhibits a number of kinases, including ROCK I (IC50 = 10.7 µM), ROCK II (IC50 = 1.9 µM), MAPK1 (IC50 = 5 µM), and PKCRK2 (IC50 = 4 µM). Weaker inhibitor of PKC (IC50 = 425 µM) and MLCK (IC50 = 95 µM) .

Storage Temperature:

Store at or below -20°C. Solid form is stable at least 12 months from date of receipt, when stored a

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