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I-BET762

Catalogue number:
CAY10676-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£42.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1260907-17-2

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

423.9

Alternative Names:

(s)-2-(6-(4-chlorophenyl)-8-methoxy-4h-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-4-yl)-n-ethylacetamide, gsk525762a

Product Description:

A synthetic compound which interacts with BET proteins with high-affinity (Kd = 32.5-42.5 nM); disrupts binding of BET proteins with acetylated histones, suppressing the expression of specific inflammatory genes involved in sepsis and endotoxic shock

Storage Temperature:

-20°C

CAY10676-1 mg: I-BET762
CAY10676-1 mg: I-BET762
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