www.bioscience.co.uk
Sales & Support: +44 (0)1223 316 855

*

GNE-7915

Catalogue number:
CAY16252-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£121.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1351761-44-8

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

443.4

Alternative Names:

[4-[[4-(ethylamino)-5-(trifluoromethyl)-2-pyrimidinyl]amino]-2-fluoro-5-methoxyphenyl]-4-morpholinyl-methanone

Product Description:

A selective, brain-penetrable LRRK2 inhibitor (Kis = 2 and 18.7 nM in biochemical and cell-based assays, respectively); inhibits LRRK2 Ser1292 autophosphorylation in BAC transgenic mice expressing human LRRK2 protein with the G2019S Parkinson’s disease mutation (IC50 = 20 nM in vivo)

Storage Temperature:

-20°C

CAY16252-5 mg: GNE-7915
CAY16252-5 mg: GNE-7915
Details Cat number & supplier Size Price
GNE-7915 CAY16252-10 mg · Cayman Chemical
CAY16252-10 mg
Cayman Chemical
10 mg £216.00
10 mg
view
GNE-7915 CAY16252-50 mg · Cayman Chemical
CAY16252-50 mg
Cayman Chemical
50 mg £710.00
50 mg
view
Dapivirine CAY16247-5 mg · Cayman Chemical
CAY16247-5 mg
Cayman Chemical
5 mg £223.00
5 mg
view
GNF-5 CAY16254-10 mg · Cayman Chemical
CAY16254-10 mg
Cayman Chemical
10 mg £85.00
10 mg
view
Dapivirine CAY16247-25 mg · Cayman Chemical
CAY16247-25 mg
Cayman Chemical
25 mg £691.00
25 mg
view
GNF-5 CAY16254-25 mg · Cayman Chemical
CAY16254-25 mg
Cayman Chemical
25 mg £140.00
25 mg
view
Dapivirine CAY16247-10 mg · Cayman Chemical
CAY16247-10 mg
Cayman Chemical
10 mg £361.00
10 mg
view
GNF-5 CAY16254-5 mg · Cayman Chemical
CAY16254-5 mg
Cayman Chemical
5 mg £48.00
5 mg
view
Dapivirine CAY16247-1 mg · Cayman Chemical
CAY16247-1 mg
Cayman Chemical
1 mg £58.00
1 mg
view
GNF-5 CAY16254-50 mg · Cayman Chemical
CAY16254-50 mg
Cayman Chemical
50 mg £253.00
50 mg
view