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BIX02188

Catalogue number:
CAY16238-10 mg
Supplier:
Size:
10 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£361.00 Estimated delivery Wed 7 Aug
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

334949-59-6

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

412.5

Alternative Names:

(3z)-3-[[[3-[(dimethylamino)methyl]phenyl]amino]phenylmethylene]-2,3-dihydro-2-oxo-1h-indole-6-carboxamide

Product Description:

A potent inhibitor of MEK5 (IC50 = 4.3 nM) and moderate inhibitor of ERK5 and TGFβR1 (IC50s = 810 and 1800 nM, respectively)

Storage Temperature:

-20°C

CAY16238-10 mg: BIX02188
CAY16238-10 mg: BIX02188
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