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MK-0457

Catalogue number:
CAY13600-250 mg
Supplier:
Size:
250 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£708.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

639089-54-6

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

464.6

Alternative Names:

n-[4-[[4-(4-methyl-1-piperazinyl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]-2-pyrimidinyl]thio]phenyl]-cyclopropanecarboxamide, tozasertib, vx-680

Product Description:

A potent pan-Aurora kinase inhibitor that favors Aurora A (Ki = 0.6 nM) over Aurora B (Ki = 18 nM) or Aurora C (Ki = 4.6 nM); inhibits proliferation of clear cell renal carcinoma (IC50 = 2/M phase

Storage Temperature:

-20°C

CAY13600-250 mg: MK-0457
CAY13600-250 mg: MK-0457
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