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EPZ004777 (formate)

Catalogue number:
CAY16173-10 mg
Supplier:
Size:
10 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£373.00 Estimated delivery Fri 9 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

585.7

Alternative Names:

7-[5-deoxy-5-[[3-[[[[4-(1,1-dimethylethyl)phenyl]amino]carbonyl]amino]propyl](1-methylethyl)amino]-β-d-ribofuranosyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine, monoformic acid

Product Description:

A potent DOT1L inhibitor (IC50 = 400 pM) that selectively kills (MLL) cells in vitro and prolongs survival in an MLL xenograft mouse model; accelerates the reprogramming of somatic cells into induced pluripotent stem cells

Storage Temperature:

-20°C

CAY16173-10 mg: EPZ004777 (formic acid s
CAY16173-10 mg: EPZ004777 (formic acid salt)
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