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PF-4800567

Catalogue number:
CAY19171-5 mg
Supplier:
Size:
5 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£185.00 Estimated delivery Fri 9 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1188296-52-7

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

359.8

Alternative Names:

3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine

Product Description:

A selective inhibitor of casein kinase 1ε (CK1ε; IC50 = 32 nM) with greater than 20-fold selectivity over CK1δ; blocks CK1ε-mediated PER3 nuclear localization and PER2 degradation, both of which are proteins important for maintaining circadian rhythms in cells

Storage Temperature:

-20°C

CAY19171-5 mg: PF-4800567
CAY19171-5 mg: PF-4800567
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