£367.00
Estimated delivery Fri 9 Aug
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
942183-80-4
Purity:
≥95%
Formulation:
A crystalline solid
Molecular Weight:
587.7
Alternative Names:
(3r)-1-[2-oxo-2-[4-[4-(2-pyrimidinyl)phenyl]-1-piperazinyl]ethyl]-n-[3-(4-pyridinyl)-1h-indazol-5-yl]-3-pyrrolidinecarboxamide
- Data sheet: View or download
- MSDS: View or download
Product Description:
A potent, selective inhibitor of ERK1 and ERK2 (IC50s = 4 and 1 nM, respectively); has nanomolar cytotoxicity in tumor cells with mutations in BRAF, NRAS, or KRAS; effective in vivo, inducing regression of xenograft tumors in mice
Storage Temperature:
-20°C
