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CP 724,714

Catalogue number:
CAY19172-5 mg
Supplier:
Size:
5 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£224.00 Estimated delivery Fri 9 Aug
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

383432-38-0

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

469.5

Alternative Names:

2-methoxy-n-[(2e)-3-[4-[[3-methyl-4-[(6-methyl-3-pyridinyl)oxy]phenyl]amino]-6-quinazolinyl]-2-propen-1-yl]-acetamide

Product Description:

A selective inhibitor of HER2/ErbB2 (IC50 = 10 nM); inhibits the proliferation of ErbB2-amplified cells, including BT474 and SK-BR-3 (IC50s = 0.25 and 0.95 µM, respectively) and demonstrates antitumor activity in various human tumor xenograft models

Storage Temperature:

-20°C

CAY19172-5 mg: CP 724,714
CAY19172-5 mg: CP 724,714
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