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EPZ011989

Catalogue number:
CAY19161-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
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  • Rest of World
£296.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1598383-40-4

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

605.8

Alternative Names:

n-[(1,2-dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-3-[ethyl[trans-4-[(2-methoxyethyl)methylamino]cyclohexyl]amino]-2-methyl-5-[3-(4-morpholinyl)-1-propyn-1-yl]-benzamide

Product Description:

A selective, orally bioavailable EZH2 inhibitor with Ki values that are less than 3 nM for wild type and Tyr646 mutant of EZH2; demonstrates significant tumor growth inhibition in a mouse xenograft model of human B cell lymphoma

Storage Temperature:

-20°C

CAY19161-1 mg: EPZ011989
CAY19161-1 mg: EPZ011989
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