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GSK2879552

Catalogue number:
CAY19403-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£142.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1401966-69-5

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

364.5

Alternative Names:

4-[[4-[[[(1r,2s)-2-phenylcyclopropyl]amino]methyl]-1-piperidinyl]methyl]-benzoic acid

Product Description:

A selective, orally bioavailable, mechanism-based inactivator of LSD1/CoREST activity; enhances H3K4 methylation, increasing the expression of tumor-suppressor genes and preventing growth of AML cell lines (EC50s = 2-240 nM)

Storage Temperature:

-20°C

CAY19403-5 mg: GSK2879552
CAY19403-5 mg: GSK2879552
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