CL 387,785
Catalogue number:
CAY19081-1 mg
Supplier:
Size:
1 mg
Product is available in:
£48.00
Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
194423-06-8
Purity:
≥95%
Formulation:
A crystalline solid
Molecular Weight:
381.2
Alternative Names:
n-[4-[(3-bromophenyl)amino]-6-quinazolinyl]-2-butynamide, ekb-785, eki-785, way-eki-785
- Data sheet: View or download
- MSDS: View or download
Product Description:
A potent, irreversible inhibitor of EGFR kinase activity (IC50 = 370 pM); halts cell cycling in cells that overexpress EGFR or c-ErbB2 (IC50s = 31-125 nM); profoundly blocks the growth of EGFR-overexpressing tumors in nude mice when given orally at 80 mg/kg/day for 10 days
Storage Temperature:
-20°C