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CL 387,785

Catalogue number:
CAY19081-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£48.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

194423-06-8

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

381.2

Alternative Names:

n-[4-[(3-bromophenyl)amino]-6-quinazolinyl]-2-butynamide, ekb-785, eki-785, way-eki-785

Product Description:

A potent, irreversible inhibitor of EGFR kinase activity (IC50 = 370 pM); halts cell cycling in cells that overexpress EGFR or c-ErbB2 (IC50s = 31-125 nM); profoundly blocks the growth of EGFR-overexpressing tumors in nude mice when given orally at 80 mg/kg/day for 10 days

Storage Temperature:

-20°C

CAY19081-1 mg: CL 387,785
CAY19081-1 mg: CL 387,785
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