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SCH 772984

Catalogue number:
CAY19166-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£48.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

942183-80-4

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

587.7

Alternative Names:

(3r)-1-[2-oxo-2-[4-[4-(2-pyrimidinyl)phenyl]-1-piperazinyl]ethyl]-n-[3-(4-pyridinyl)-1h-indazol-5-yl]-3-pyrrolidinecarboxamide

Product Description:

A potent, selective inhibitor of ERK1 and ERK2 (IC50s = 4 and 1 nM, respectively); has nanomolar cytotoxicity in tumor cells with mutations in BRAF, NRAS, or KRAS; effective in vivo, inducing regression of xenograft tumors in mice

Storage Temperature:

-20°C

CAY19166-1 mg: SCH 772984
CAY19166-1 mg: SCH 772984
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