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HI TOPK 032

Catalogue number:
CAY19815-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£45.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

487020-03-1

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

369.4

Alternative Names:

n-(12-cyanoindolizino[2,3-b]quinoxalin-2-yl)-2-thiophenecarboxamide

Product Description:

An inhibitor of TOPK (IC50 = ~2 µM), Chk1 (IC50 = 9.6 µM), and MEK1 (40% inhibition at 5 µM); decreases the growth of colon cancer and glioma initiating cells in vitro and suppresses tumor growth in vivo

Storage Temperature:

-20°C

CAY19815-1 mg: HI TOPK 032
CAY19815-1 mg: HI TOPK 032
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