10074-G5
Catalogue number:
CAY17408-10 mg
Supplier:
Size:
10 mg
Product is available in:
£142.00
Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
413611-93-5
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Weight:
332.3
Alternative Names:
n-[1,1'-biphenyl]-2-yl-7-nitro-2,1,3-benzoxadiazol-4-amine
- Data sheet: View or download
- MSDS: View or download
Product Description:
A c-Myc inhibitor that binds to and distorts the bHLH-ZIP domain of c-Myc (Kd = 2.8 µM), thereby inhibiting c-Myc/Max heterodimer formation and inhibiting its transcriptional activity (IC50 = 146 µM); cytotoxic to c-Myc-overexpressing cells lines (IC50s = 15.6 and 13.5 µM for Daudi Burkitt lymphoma cells and HL60 promyelocytic leukemia cells, respectively)
Storage Temperature:
-20°C