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PD 168368

Catalogue number:
CAY17920-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£315.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

204066-82-0

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

554.6

Alternative Names:

(αs)-α-methyl-α-[[[(4-nitrophenyl)amino]carbonyl]amino]-n-[[1-(2-pyridinyl)cyclohexyl]methyl]-1h-indole-3-propanamide

Product Description:

A competitive, selective antagonist of NMB receptors (Kis = 15-45 nM for rat and human receptors expressed in various cell lines); blocks the elevation of intracellular calcium and release of inositol phosphate induced by NMB in cells expressing NMB receptors

Storage Temperature:

-20°C

CAY17920-5 mg: PD 168368
CAY17920-5 mg: PD 168368
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