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HG-10-102-01

Catalogue number:
CAY20049-10 mg
Supplier:
Size:
10 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£247.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1351758-81-0

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

377.8

Alternative Names:

[4-[[5-chloro-4-(methylamino)-2-pyrimidinyl]amino]-3-methoxyphenyl]-4-morpholinyl-methanone

Product Description:

An inhibitor of LRRK2 (IC50 = 20.3 nM); also inhibits G2019S, A2016T, and [G2019S+A2016T] mutants of LRRK2 (IC50s = 3.2, 153, and 95.9 nM, respectively); brain penetrant and inhibits Ser910 and Ser935 phosphorylation of both wild-type and G2019S mutant LRRK2

Storage Temperature:

-20°C

CAY20049-10 mg: HG-10-102-01
CAY20049-10 mg: HG-10-102-01
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