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SGI-7079

Catalogue number:
CAY20111-10 mg
Supplier:
Size:
10 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£315.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1239875-86-5

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

455.5

Alternative Names:

3-[2-[[3-fluoro-4-(4-methyl-1-piperazinyl)phenyl]amino]-5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl]-benzeneacetonitrile

Product Description:

An Axl kinase inhibitor; inhibits proliferation of inflammatory breast cancer cells (IC50s = 0.43 and 0.15 µM for SUM149 and KPL-4 cells, respectively); synergistically increases the potency of erlotinib on EGFR inhibition; dose-dependently inhibits tumor growth in a mouse xenograft model of non-small cell lung cancer

Storage Temperature:

-20°C

CAY20111-10 mg: SGI-7079
CAY20111-10 mg: SGI-7079
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