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Epacadostat

Catalogue number:
CAY19875-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£42.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1204669-58-8

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

438.2

Alternative Names:

[c(z)]-4-[[2-[(aminosulfonyl)amino]ethyl]amino]-n-(3-bromo-4-fluorophenyl)-n'-hydroxy-1,2,5-oxadiazole-3-carboximidamide, incb024360

Product Description:

A selective IDO1 inhibitor (IC50 = 7.1 nM in HeLa cells); promotes T and natural killer-cell growth, increases IFN-γ production, and reduces conversion to Treg-like cells in a coculture system of human allogeneic lymphocytes with either dendritic cells or tumor cells; inhibits tumor growth in tumor-bearing mice in a lymphocyte-dependent manner

Storage Temperature:

-20°C

CAY19875-1 mg: Epacadostat
CAY19875-1 mg: Epacadostat
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