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Uprosertib

Catalogue number:
CAY19904-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£42.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1047634-65-0

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

429.2

Alternative Names:

n-[(1s)-2-amino-1-[(3,4-difluorophenyl)methyl]ethyl]-5-chloro-4-(4-chloro-1-methyl-1h-pyrazol-5-yl)-2-furancarboxamide, gsk2141795, gsk795

Product Description:

A selective, orally bioavailable inhibitor of Akt (IC50s = 180, 328, and 38 nM for Akt1, Akt2, and Akt3, respectively); preferentially inhibits the proliferation of human cancer cells lines with Akt pathway activation via PI3K/PTEN mutation or loss

Storage Temperature:

-20°C

CAY19904-1 mg: Uprosertib
CAY19904-1 mg: Uprosertib
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