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MI-136

Catalogue number:
CAY19245-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£48.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1628316-74-4

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

470.5

Alternative Names:

5-[[4-[[6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl]amino]-1-piperidinyl]methyl]-1h-indole-2-carbonitrile

Product Description:

An inhibitor of the menin-MLL interaction (IC50 = 31 nM; Kd = 23.6 nM); blocks AR signaling, inhibiting the growth of castration-resistant tumors in mice

Storage Temperature:

-20°C

CAY19245-1 mg: MI-136
CAY19245-1 mg: MI-136
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