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INCB 28060

Catalogue number:
CAY20056-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£115.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1029712-80-8

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

412.4

Alternative Names:

2-fluoro-n-methyl-4-[7-(6-quinolinylmethyl)imidazo[1,2-b][1,2,4]triazin-2-yl]-benzamide, capmatinib, inc 280

Product Description:

An inhibitor of HGFR potently blocking in vitro kinase activity (IC50 = 0.13 nM) as well as constitutive or HGF-stimulated activity in cells (IC50 values range from 0.3 to 1.1 nM); orally bioavailable, inhibiting the growth of HGFR-dependent tumors in mice

Storage Temperature:

-20°C

CAY20056-5 mg: INCB 28060
CAY20056-5 mg: INCB 28060
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