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Pelitinib

Catalogue number:
CAY15627-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£58.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

257933-82-7

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

467.9

Alternative Names:

n-[4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2e-butenamide, ekb-569

Product Description:

A cyanoquinoline that irreversibly inhibits the receptor tyrosine kinases EGFR (IC50 = 39 nM) and HER2 (IC50 = 1.2 µM); disrupts Akt and MAPK pathways, inducing apoptosis and suppressing the growth of tumor cell lines

Storage Temperature:

-20°C

CAY15627-1 mg: Pelitinib
CAY15627-1 mg: Pelitinib
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