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GDC-0032

Catalogue number:
CAY17387-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£151.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1282512-48-4

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

460.5

Alternative Names:

4-[5,6-dihydro-2-[3-methyl-1-(1-methylethyl)-1h-1,2,4-triazol-5-yl]imidazo[1,2-d][1,4]benzoxazepin-9-yl]-α,α-dimethyl-1h-pyrazole-1-acetamide, ​taselisib

Product Description:

A potent inhibitor of PI3K isoforms α, δ, and γ (IC50s = 0.28, 0.12, and 0.97 nM, respectively) that is 31 times less potent at PI3Kβ; has increased potency in cancer cell lines harboring PIK3CA-activating alterations, and is effective in vivo

Storage Temperature:

-20°C

CAY17387-5 mg: GDC-0032
CAY17387-5 mg: GDC-0032
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