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PHA-848125

Catalogue number:
CAY21474-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£175.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

802539-81-7

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

460.6

Alternative Names:

4,5-dihydro-n,1,4,4-tetramethyl-8-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide, milciclib

Product Description:

An ATP-competitive inhibitor of Cdks that most potently inhibits Cdk2/cyclin A (IC50 = 45 nM); more than 3-fold less potent at Cdks 1, 3, 4, 5, and 7

Storage Temperature:

-20°C

CAY21474-5 mg: PHA-848125
CAY21474-5 mg: PHA-848125
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