AC-262536
Catalogue number:
CAY31598-5 mg
Supplier:
Size:
5 mg
Product is available in:
£251.00
Estimated delivery Tue 6 Aug
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
870888-46-3
Purity:
≥98%
Formulation:
A solid
Molecular Weight:
278.4
Alternative Names:
4-[(3-endo)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-naphthalenecarbonitrile
- Data sheet: View or download
- MSDS: View or download
Product Description:
A SARM (Ki = 5.01 nM); an androgen receptor partial agonist (EC50 = 1.58 nM in a luciferase assay); selective for the androgen receptor over a panel of 47 additional human nuclear receptors at 10 µM; inhibits dihydroxytestosterone-induced proliferation of LNCaP prostate cancer cells at 0.1 and 1 µM; reduces plasma luteinizing hormone levels and increases levator ani muscle weight in castrated rats at 3, 10, and 30 mg/kg; exhibits smaller increases in prostate gland and seminal vesicle weight compared with testosterone in the same model
Storage Temperature:
-20°C