£371.00
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
625092-10-6
Purity:
≥98%
Formulation:
A solid
Molecular Weight:
1651.3
Alternative Names:
n-acetyl-3-(2-naphthalenyl)-d-alanyl-4-chloro-d-phenylalanyl-3-(3-pyridinyl)-d-alanyl-l-seryl-n6-(3-pyridinylcarbonyl)-l-lysyl-n6-(3-pyridinylcarbonyl)-d-lysyl-l-leucyl-n6-(1-methylethyl)-l-lysyl-l-prolyl-d-alaninamide, monoacetate
- Data sheet: View or download
- MSDS: View or download
Product Description:
A GnRHR antagonist; inhibits GnRH-induced secretion of LH, FSH, and gonadotropin in isolated rat pituitary cells (0.001-1,000 nM) but does not induce histamine release in isolated rat mast cells (EC50 = >300 µg/ml); reduces serum LH and FSH levels in orchidectomized cynomolgus monkeys at 250 µg/kg; inhibits ovulation in rats at 2 µg/animal; reduces the intensity and duration of haloperidol-induced catalepsy at 10 µg/animal
Storage Temperature:
-20°C