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Alflutinib (mesylate)

Catalogue number:
CAY31473-5 mg
Supplier:
Size:
5 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£157.00 Estimated delivery Fri 9 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

2130958-55-1

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

664.7

Alternative Names:

n-[2-[[2-(dimethylamino)ethyl]methylamino]-5-[[4-(1-methyl-1h-indol-3-yl)-2-pyrimidinyl]amino]-6-(2,2,2-trifluoroethoxy)-3-pyridinyl]-2-propenamide, monomethanesulfonate, ast2818

Product Description:

An inhibitor of mutant EGFRs; selective for EGFRL858R, EGFRG719X, EGFRL858R, EGFRL861A, and EGFRT790M mutant EGFRs over wild-type EGFR; reduces tumor growth in an EGFRL858R and EGFRT790M-expressing LU1868 NSCLC PDX mouse model at 10 and 30 mg/kg

Storage Temperature:

-20°C

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